Molecule Details
InChIKeyPNSVJQJVGCLXPD-UHFFFAOYSA-N
Compound Name4-tert-butyl-N-(6-oxo-1H-pyridin-3-yl)-2-[6-(trifluoromethyl)pyridin-3-yl]oxybenzamide
Canonical SMILESCC(C)(C)c1ccc(C(=O)Nc2ccc(=O)[nH]c2)c(Oc2ccc(C(F)(F)F)nc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.19
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y5Y9 SCN10A Homo sapiens Human PF00520 PF24609 PF06512 6.2 IC50 ChEMBL;BindingDB
Q9UQD0 SCN8A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 6.2 IC50 ChEMBL;BindingDB