Molecule Details
InChIKeyPNAQMBCCITXUCG-UHFFFAOYSA-N
Compound NameN-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-[6-(dimethylamino)-3-pyridinyl]acetamide
Canonical SMILESCN(C)c1ccc(CC(=O)Nc2ccn(Cc3ccc(F)c(F)c3)n2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P0X4 CACNA1I Homo sapiens Human PF00520 8.4 IC50 ChEMBL;BindingDB
O43497 CACNA1G Homo sapiens Human PF00520 7.9 IC50 ChEMBL;BindingDB
O95180 CACNA1H Homo sapiens Human PF00520 7.3 IC50 ChEMBL;BindingDB