Molecule Details
InChIKeyPMXQIBXLHFWGQH-UHFFFAOYSA-O
Compound Name2,4,6-Trimethyl-1-[(5-sulfamoyl-[1,3,4]thiadiazol-2-ylcarbamoyl)-methyl]-pyridinium; perchlorate
Canonical SMILESCc1cc(C)[n+](CC(=O)Nc2nnc(S(N)(=O)=O)s2)c(C)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.51
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 8.0 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.0 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 6.5 Ki ChEMBL;BindingDB