Molecule Details
InChIKeyPMSCCWYCOFSMQM-UHFFFAOYSA-N
Compound NameN-[5-chloro-6-[(2-methyl-3-pyridinyl)oxy]-3-pyridinyl]-5-methyl-6-(trifluoromethyl)-2,3-dihydroindole-1-carboxamide
Canonical SMILESCc1cc2c(cc1C(F)(F)F)N(C(=O)Nc1cnc(Oc3cccnc3C)c(Cl)c1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.6
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB