Molecule Details
InChIKeyPMOWTIHVNWZYFI-AATRIKPKSA-N
Compound NameO-Coumaric Acid
Canonical SMILESO=C(O)/C=C/c1ccccc1O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Unknown
Avg pChEMBL6.92
SourceBindingDB;TTD_MultiTarget
2D Structure
2D structure
DrugBank Annotations
DrugBank ID DB01650
Drug Nametrans-2-hydroxycinnamic acid
CAS Number614-60-8
Groups experimental
ATC Codes nan
Descriptionnan

Categories: OAT3/SLC22A8 Inhibitors
Cross-references: BindingDB: 50146462 ChEBI: 18125 CHEMBL52564 ChemSpider: 553146 C01772 PDB: 2HC PubChem:637540 PubChem:46505688 ZINC: ZINC000000895911
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 Clinical TTD_MultiTarget TTD_MultiTarget
A0A045J7I4 yrdA Mycobacterium tuberculosis Pathogen 6.9 Ki BindingDB
DrugBank Target Actions (4)
Target Gene Target Name Action Type
P46072 P46072 Major NAD(P)H-flavin oxidoreductase binder targets
P00915 CA1 Carbonic anhydrase 1 inhibitor targets
P00918 CA2 Carbonic anhydrase 2 inhibitor targets
Q8TCC7 SLC22A8 Organic anion transporter 3 inhibitor transporters