Molecule Details
InChIKeyPMDUMOUXISSZED-BSYJTBJZSA-N
Compound NameN-[(S)-cyclopropyl(pyridin-2-yl)methyl]-3-[4-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)phenyl]-1H-indazole-5-carboxamide
Canonical SMILESO=C(N[C@H](c1ccccn1)C1CC1)c1ccc2[nH]nc(-c3ccc(N4C5CCC4COC5)cc3)c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.24
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P33981 TTK Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 6.4 IC50 ChEMBL
Q9NQS7 INCENP Homo sapiens Human PF03941 PF12178 6.4 IC50 ChEMBL