Molecule Details
InChIKeyPLSQYACXDKUYFC-UHFFFAOYSA-N
Compound Name(S)-5-methyl-1-(quinolin-4-ylmethyl)-3-(4-(trifluoromethylsulfonyl)phenyl)imidazolidine-2,4-dione
Canonical SMILESCc1c(O)n(-c2ccc(S(=O)(=O)C(F)(F)F)cc2)c(=O)n1Cc1ccnc2ccccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.32
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P06213 INSR Homo sapiens Human PF00757 PF17870 PF07714 PF01030 6.5 IC50 BindingDB
P08069 IGF1R Homo sapiens Human PF00757 PF07714 PF01030 6.3 IC50 BindingDB
P11712 CYP2C9 Homo sapiens Human PF00067 6.2 IC50 BindingDB