Molecule Details
InChIKeyPLQQFQYHSIBALT-UHFFFAOYSA-N
Compound Namedimethyl-{3-[(2-p-tolyl-ethylamino)-methyl]-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl}-amine
Canonical SMILESCc1ccc(CCNCC2(N(C)C)COc3ccccc3OC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.24
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P20309 CHRM3 Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB
P08172 CHRM2 Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB
P11229 CHRM1 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB