Molecule Details
InChIKeyPKQHIVDUFZWMMH-QNGWXLTQSA-N
Canonical SMILESCC(C)Oc1ccc(-c2n[nH]c3ccc(NC(=O)[C@]4(S(C)(=O)=O)CCN(CC(=O)N5CC=C(c6ccc(-c7ncn(C)n7)cc6)CC5)C4)cc23)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.09
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P28482 MAPK1 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P27361 MAPK3 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB