Molecule Details
InChIKeyPKPONRIRXFIKES-GOSISDBHSA-N
Compound Name(R)-4-[3-(3-isopropyl-phenoxy)-pyrrolidin-1-yl]-6,7-dimethoxy-quinazoline
Canonical SMILESCOc1cc2ncnc(N3CC[C@@H](Oc4cccc(C(C)C)c4)C3)c2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.38
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q14432 PDE3A Homo sapiens Human PF00233 6.4 Ki ChEMBL;BindingDB
Q13370 PDE3B Homo sapiens Human PF00233 6.3 Ki ChEMBL;BindingDB