Molecule Details
InChIKeyPKHQCKPNCMWYHX-UHFFFAOYSA-N
Compound Name1-(1-Cyclooctylpiperidin-4-yl)-3-[(6-methoxy-3-pyridinyl)amino]quinoxalin-2-one
Canonical SMILESCOc1ccc(Nc2nc3ccccc3n(C3CCN(C4CCCCCCC4)CC3)c2=O)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.78
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41145 OPRK1 Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB
Q5TC84 OGFRL1 Homo sapiens Human PF04664 6.8 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB