Molecule Details
InChIKeyPJNMAIKMKRLUIV-UHFFFAOYSA-N
Compound Name6-methoxy-3-(2-methoxy-4-pyridinyl)-N-methylpyrazolo[1,5-a]pyrimidin-5-amine
Canonical SMILESCNc1nc2c(-c3ccnc(OC)c3)cnn2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.22
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P37173 TGFBR2 Homo sapiens Human PF08917 PF07714 9.0 IC50 ChEMBL;BindingDB
P27037 ACVR2A Homo sapiens Human PF01064 PF00069 6.5 IC50 ChEMBL;BindingDB
P36897 TGFBR1 Homo sapiens Human PF01064 PF00069 PF08515 6.2 IC50 ChEMBL;BindingDB