InChIKey	PJMPHNIQZUBGLI-UHFFFAOYSA-N
Compound Name	Fentanyl
Canonical SMILES	CCC(=O)N(c1ccccc1)C1CCN(CCc2ccccc2)CC1
Clinical Status	Data-mined Candidate
Targets (Human+Pathogen)	6
Pfam Stratification	Cross-Family
Avg pChEMBL	7.89
Source	BindingDB;ChEMBL

DrugBank ID	DB00813
Drug Name	Fentanyl
CAS Number	437-38-7
Groups	approved illicit investigational vet_approved
ATC Codes	N01AH01 N02AB03 N01AH51
Description	Fentanyl, a potent opioid agonist, was developed in the 1950s to fill a need for strong and rapid analgesia.[A179542] Because of these characteristics, fentanyl is commonly used to treat chronic cancer pain or in anesthesia.[Label,L6598,L6601,L6604,L6607,L922,L6610,L6613] Fentanyl is related to othe...

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Categories: Adjuvants Adjuvants, Anesthesia Agents that produce hypertension Agents that reduce seizure threshold Analgesics Anesthetics Anesthetics, General Anesthetics, Intravenous Antidepressive Agents Bradycardia-Causing Agents Central Nervous System Agents Central Nervous System Depressants Cytochrome P-450 CYP3A Substrates Cytochrome P-450 CYP3A4 Substrates Cytochrome P-450 CYP3A7 Substrates Cytochrome P-450 Substrates Drugs that are Mainly Renally Excreted Fentanyl and fentanyl analogues High-risk opioids Narcotics Nervous System Neuraxial Anesthetics Opiate Agonists Opioid Agonist Opioid Anesthetics Opioids Opioids, Anilidopiperidine P-glycoprotein inhibitors Peripheral Nervous System Agents Phenylpiperidine opioids Piperidines Sensory System Agents Serotonergic Drugs Shown to Increase Risk of Serotonin Syndrome Serotonin Agents Serotonin Modulators

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Cross-references: BindingDB: 50008984 ChEBI: 119915 CHEMBL596 ChemSpider: 3228 Drugs Product Database (DPD): 10075 Guide to Pharmacology: 1626 IUPHAR: 1626 D00320 PDB: 7V7 PharmGKB: PA449599 PubChem:3345 PubChem:46506372 RxCUI: 4337 Therapeutic Targets Database: DAP000072 Wikipedia: Fentanyl ZINC: ZINC000002522669