Molecule Details
InChIKeyPJMOAMQVWVRXEQ-UHFFFAOYSA-N
Compound Name1-Benzyl-4-(4-methyl-5-phenyl-1H-pyrazol-3-yl)-piperidine
Canonical SMILESCc1c(C2CCN(Cc3ccccc3)CC2)n[nH]c1-c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.24
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB