Molecule Details
InChIKeyPJEKXBMIYGCRBL-UHFFFAOYSA-N
Compound Name3-cyclobutyl-1-(5-methyl-1H-indol-2-yl)imidazo[1,5-a]pyrazin-8-amine
Canonical SMILESCc1ccc2[nH]c(-c3nc(C4CCC4)n4ccnc(N)c34)cc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.4
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P22607 FGFR3 Homo sapiens Human PF21165 PF07679 PF13927 PF07714 6.6 IC50 BindingDB
P09211 GSTP1 Homo sapiens Human PF14497 PF02798 6.3 IC50 BindingDB
P11362 FGFR1 Homo sapiens Human PF07679 PF00047 PF07714 6.3 IC50 ChEMBL;BindingDB