Molecule Details
InChIKeyPITUMGJELDUJEZ-CCEZHUSRSA-N
Compound Name9-(2,6-dimethylstyryl)-N-(4-(dipropylphosphoryl)phenyl)-9H-purin-6-amine
Canonical SMILESCCCP(=O)(CCC)c1ccc(Nc2ncnc3c2ncn3/C=C/c2c(C)cccc2C)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.19
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 8.4 IC50 ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.4 pIC50 TTD_MultiTarget
P00519 ABL1 Homo sapiens Human PF08919 PF07714 PF00017 PF00018 7.8 IC50 ChEMBL;BindingDB