Molecule Details
InChIKeyPIPNMGRIVITFEC-VQCQRNETSA-N
Compound NameN-{1-(2,2-Diethyl-[1,3]dioxolan-4-yl)-2-[4-(4-trifluoromethoxy-phenoxy)-benzenesulfonyl]-ethyl}-N-hydroxy-formamide
Canonical SMILESCCC1(CC)OCC([C@@H](CS(=O)(=O)c2ccc(Oc3ccc(OC(F)(F)F)cc3)cc2)N(O)C=O)O1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.33
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 9.0 IC50 ChEMBL;BindingDB
Q9ULZ9 MMP17 Homo sapiens Human PF00045 PF00413 PF01471 8.3 pIC50 TTD_MultiTarget
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 7.7 pIC50 TTD_MultiTarget