Molecule Details
InChIKeyPIMQWRZWLQKKBJ-GOSISDBHSA-N
Compound Name2-[(2R)-1-[3-ethyl-7-[(1-oxidopyridin-1-ium-3-yl)methylamino]pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-2-yl]ethanol
Canonical SMILESCCc1cnn2c(NCc3ccc[n+]([O-])c3)cc(N3CCCC[C@@H]3CCO)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL8.73
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 9.0 IC50 ChEMBL
Q00535 CDK5 Homo sapiens Human PF00069 9.0 IC50 ChEMBL
P06493 CDK1 Homo sapiens Human PF00069 8.5 IC50 ChEMBL
P50750 CDK9 Homo sapiens Human PF00069 8.4 IC50 ChEMBL