Molecule Details
InChIKeyPHZQLNMARSMWBL-LJDCWIOTSA-N
Canonical SMILES[N][C][C][C][C][C@@H]([N]C(=O)[C][C][C][C][C][N]C(=O)[C@H]1O[C@@H](n2cnc3c([N])ncnc32)[C@H]([O])[C@@H]1[O])C(=O)[N][C][C][C][C][C]C(=O)[N][C@H]([C][C][C]N=C([N])[N])C(=O)[N][C@H]([C][C][C]N=C([N])[N])C(=O)[N][C@H]([C][C][C]N=C([N])[N])C(=O)[N][C@H]([C][C][C]N=C([N])[N])C(=O)[N][C@H]([C][C][C]N=C([N])[N])C(=O)[N][C@H]([C][C][C]N=C([N])[N])C([N])=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.26
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O75116 ROCK2 Homo sapiens Human PF25346 PF00069 PF08912 10.7 Kd BindingDB
Q9Y243 AKT3 Homo sapiens Human PF00169 PF00069 PF00433 7.8 IC50 BindingDB