Molecule Details
InChIKeyPHVWYDDIUNHCKW-UHFFFAOYSA-N
Compound Name3-(1H-Imidazol-1-yl)-6-{4-[2-(trifluoromethyl)phenoxy]piperidin-1-yl}pyridazine
Canonical SMILESFC(F)(F)c1ccccc1OC1CCN(c2ccc(-n3ccnc3)nn2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.46
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P10635 CYP2D6 Homo sapiens Human PF00067 6.5 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.4 IC50 ChEMBL;BindingDB