Molecule Details
InChIKeyPHBGFWHJUVWHAA-UHFFFAOYSA-N
Compound Name2,2,2-Trifluoro-1-[5-(quinoxalin-6-yl)thiophen-2-yl]ethanone
Canonical SMILESO=C(c1ccc(-c2ccc3nccnc3c2)s1)C(F)(F)F
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.63
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 7.8 IC50 ChEMBL;BindingDB
Q02161 RHD Homo sapiens Human PF00909 6.0 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 6.0 pIC50 TTD_MultiTarget