Molecule Details
InChIKeyPGVYYPZKXKGBLD-JKSUJKDBSA-N
Compound Name(3R,4R)-N-hydroxy-4-[[4-[[2-(trifluoromethyl)benzimidazol-1-yl]methyl]benzoyl]amino]oxane-3-carboxamide
Canonical SMILESO=C(N[C@@H]1CCOC[C@@H]1C(=O)NO)c1ccc(Cn2c(C(F)(F)F)nc3ccccc32)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.45
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P78536 ADAM17 Homo sapiens Human PF16698 PF00200 PF13574 6.9 IC50 ChEMBL;BindingDB
Q9UNA0 ADAMTS5 Homo sapiens Human PF17771 PF19236 PF05986 PF01421 PF19030 PF00090 6.0 Ki ChEMBL