Molecule Details
InChIKeyPGUYNSUWECOWIP-BUSXIPJBSA-N
Compound NameN-((S)-1-Carbamimidoyl-2-hydroxy-piperidin-3-yl)-2-(2-methyl-6-oxo-5-phenylmethanesulfonylamino-6H-pyrimidin-1-yl)-acetamide
Canonical SMILESCc1ncc(NS(=O)(=O)Cc2ccccc2)c(=O)n1CC(=O)N[C@H]1CCCN(C(=N)N)C1O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.16
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 8.6 IC50 ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 6.8 IC50 ChEMBL;BindingDB
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 6.0 IC50 ChEMBL;BindingDB