Molecule Details
InChIKeyPGTDWVFHKGDQFC-KLSDWBHSSA-N
Canonical SMILESCC[C@H](C)[C@@H]1C(=O)O[C@H]1C(=O)N[C@H](C(=O)N[C@@H](COCc1ccccc1)C(=O)OCc1ccccc1)C(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P28074 PSMB5 Homo sapiens Human PF00227 8.5 IC50 ChEMBL;BindingDB
P28062 PSMB8 Homo sapiens Human PF00227 8.0 IC50 ChEMBL;BindingDB