Molecule Details
InChIKeyPGAPJRVJNZPHAS-ABAIWWIYSA-N
Compound Name2,5-difluoro-4-[(1S,2R)-2-(2-methylpyrazol-3-yl)cyclopentyl]oxy-N-(1,3-thiazol-2-yl)benzenesulfonamide
Canonical SMILESCn1nccc1[C@H]1CCC[C@@H]1Oc1cc(F)c(S(=O)(=O)Nc2nccs2)cc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O60939 SCN2B Homo sapiens Human PF07686 7.5 IC50 ChEMBL;BindingDB
Q07699 SCN1B Homo sapiens Human PF07686 7.5 IC50 ChEMBL
Q15858 SCN9A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 7.5 IC50 ChEMBL;BindingDB