Molecule Details
InChIKeyPFHKAGAZRDERTK-OAQYLSRUSA-N
Compound NameN-[(1s)-2-Hydroxy-1-Phenylethyl]-4-[5-Methyl-2-(Phenylamino)pyrimidin-4-Yl]-1h-Pyrrole-2-Carboxamide
Canonical SMILESCc1cnc(Nc2ccccc2)nc1-c1c[nH]c(C(=O)N[C@H](CO)c2ccccc2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL8.04
SourceBindingDB;ChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P28482 MAPK1 Homo sapiens Human PF00069 8.4 Ki BindingDB
P49841 GSK3B Homo sapiens Human PF00069 8.2 Ki BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.8 Ki ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.8 pIC50 TTD_MultiTarget