Molecule Details
InChIKeyPFEBJWBMYVVIJO-UHFFFAOYSA-N
Compound Name2-Methyl-5-[2-[4-[[3-(1-methylpiperidin-4-yl)phenyl]methyl]piperidin-1-yl]ethoxy]quinoline
Canonical SMILESCc1ccc2c(OCCN3CCC(Cc4cccc(C5CCN(C)CC5)c4)CC3)cccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 9.7 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB