Molecule Details
InChIKeyPFAXMIALVXBXEB-UHFFFAOYSA-N
Compound Name2-(2,6-Difluorobenzyl)-8-(2-(dimethylamino) pyridin-4-yl)-7-(4-fluorophenyl)-[l,2,4]triazolo [l,5-c]pyrmidin-5-amine
Canonical SMILESCN(C)c1cc(-c2c(-c3ccc(F)cc3)nc(N)n3nc(Cc4c(F)cccc4F)nc23)ccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 10.0 IC50 ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 9.1 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 8.6 IC50 ChEMBL;BindingDB