Molecule Details
InChIKeyPETRMFAIRNHKGK-UHFFFAOYSA-N
Compound NameN-[3-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine
Canonical SMILESCN1CCN(c2cccc(Nc3nccc(-c4cn(C)c5ncccc45)n3)c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 7.6 Ki ChEMBL;BindingDB
P24864 CCNE1 Homo sapiens Human PF02984 PF00134 6.0 Ki ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 6.0 Ki ChEMBL;BindingDB