Molecule Details
InChIKeyPETMAGJXWYMKMA-UHFFFAOYSA-N
Canonical SMILESCc1nc(OCC2(F)CCOCC2)sc1S(=O)(=O)NC(=O)c1ccc(N2CCN(CC3=C(c4ccc(Cl)cc4)CC(C)(C)CC3)CC2)cc1Oc1cccc2[nH]cnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.76
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P10415 BCL2 Homo sapiens Human PF00452 PF02180 8.8 Ki ChEMBL;BindingDB
Q07817 BCL2L1 Homo sapiens Human PF00452 PF02180 8.8 Ki ChEMBL;BindingDB