Molecule Details
InChIKeyPELASOGQJSUMMW-GOSISDBHSA-N
Compound Name4-(((R)-2-((1H-indol-3-yl)methyl)-3,6-dioxopiperazin-1-yl)methyl)-N-hydroxybenzamide
Canonical SMILESO=C(NO)c1ccc(CN2C(=O)CNC(=O)[C@H]2Cc2c[nH]c3ccccc23)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.96
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q02161 RHD Homo sapiens Human PF00909 7.0 pIC50 TTD_MultiTarget
Q92769 HDAC2 Homo sapiens Human PF00850 7.0 pIC50 TTD_MultiTarget
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 7.0 IC50 ChEMBL;BindingDB