Molecule Details
InChIKeyPDRMZIBUTGMDNS-UHFFFAOYSA-N
Canonical SMILESCc1ccn2c(-c3ccc4cccc(OCC(C)(C)CN)c4n3)nnc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.93
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.1 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB