Molecule Details
InChIKeyPDJZASCRQRBYQS-UHFFFAOYSA-N
Canonical SMILESO=C(NCc1ccccc1)c1cc(-c2n[nH]cc2-c2cccc(Cl)c2)c[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB07010
Drug NameN-BENZYL-4-[4-(3-CHLOROPHENYL)-1H-PYRAZOL-3-YL]-1H-PYRROLE-2-CARBOXAMIDE
CAS Numbernan
Groups experimental
ATC Codes nan
Descriptionnan

Cross-references: BindingDB: 225377 CHEMBL220320 ChemSpider: 22376242 PDB: 33A PubChem:10134160 PubChem:99443481 ZINC: ZINC000020149027
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P28482 MAPK1 Homo sapiens Human PF00069 7.1 Ki ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.3 Ki ChEMBL;BindingDB
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P28482 MAPK1 Mitogen-activated protein kinase 1 binder targets
P53779 MAPK10 Mitogen-activated protein kinase 10 binder targets