Molecule Details
InChIKeyPDGBJOHNOOKHMI-HSZRJFAPSA-N
Compound NamePyrimidylpyrrole, 9c
Canonical SMILESCCc1ccccc1Nc1ncc(C)c(-c2c[nH]c(C(=O)N[C@H](CO)c3ccccc3)c2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.11
SourceBindingDB;ChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28482 MAPK1 Homo sapiens Human PF00069 8.5 Ki ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.7 pIC50 TTD_MultiTarget
P49841 GSK3B Homo sapiens Human PF00069 6.1 Ki BindingDB