Molecule Details
InChIKeyPCXIRNWRIJAIPA-UHFFFAOYSA-N
Compound Name3-(2,5-dioxopyrrolidin-1-yl)-N-(4-sulfamoylphenyl)benzamide
Canonical SMILESNS(=O)(=O)c1ccc(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16790 CA9 Homo sapiens Human PF00194 7.7 IC50 ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 7.5 IC50 ChEMBL;BindingDB
P00915 CA1 Homo sapiens Human PF00194 6.9 IC50 ChEMBL;BindingDB