Molecule Details
InChIKeyPBTHEXRSPYUHQA-UHFFFAOYSA-N
Compound NameN-[4-(4,5-Dihydro-2H-9-thia-1,2,6-triaza-cyclopenta[e]azulene-6-carbonyl)-phenyl]-2-methyl-benzamide
Canonical SMILESCc1ccccc1C(=O)Nc1ccc(C(=O)N2CCc3c[nH]nc3-c3sccc32)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30518 AVPR2 Homo sapiens Human PF00001 6.9 IC50 ChEMBL;BindingDB
P37288 AVPR1A Homo sapiens Human PF00001 PF08983 6.6 IC50 ChEMBL;BindingDB