Molecule Details
InChIKeyPBFKMRLPTUCFLU-UHFFFAOYSA-N
Compound Name4-[5-(2-Methoxyphenoxy)-2-morpholin-4-yl-6-[(5-propan-2-yl-2-pyridinyl)sulfonylamino]pyrimidin-4-yl]oxybut-2-ynyl pyridine-2-carboxylate
Canonical SMILESCOc1ccccc1Oc1c(NS(=O)(=O)c2ccc(C(C)C)cn2)nc(N2CCOCC2)nc1OCC#CCOC(=O)c1ccccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.19
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P25101 EDNRA Homo sapiens Human PF00001 9.0 IC50 ChEMBL;BindingDB
P24530 EDNRB Homo sapiens Human PF00001 7.4 IC50 ChEMBL;BindingDB