Molecule Details
InChIKeyPBCRELBKGRVORN-DFVFADGESA-N
Compound NameH-Dip-Cys(1)-Tyr-D-Trp-Lys-Val-Cys(1)-Dip-NH2
Canonical SMILESCC(C)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@@H](NC(=O)[C@@H](N)C(c2ccccc2)c2ccccc2)CSSC[C@@H](C(=O)N[C@H](C(N)=O)C(c2ccccc2)c2ccccc2)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30874 SSTR2 Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P35346 SSTR5 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB