Molecule Details
InChIKeyPAIPLWPUQXJMMT-UHFFFAOYSA-N
Compound NameN-[4-[[3-[[5-(trifluoromethyl)-2-pyridyl]oxy]phenyl]methylene]cyclohexyl]-pyridine-3-carboxamide
Canonical SMILESO=C(NC1CCC(=Cc2cccc(Oc3ccc(C(F)(F)F)cn3)c2)CC1)c1cccnc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL8.64
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P08684 CYP3A4 Homo sapiens Human PF00067 9.0 IC50 ChEMBL
O00519 FAAH Homo sapiens Human PF01425 8.7 IC50 ChEMBL
P11712 CYP2C9 Homo sapiens Human PF00067 8.6 IC50 ChEMBL
P33261 CYP2C19 Homo sapiens Human PF00067 8.3 IC50 ChEMBL