Molecule Details
InChIKeyPABWXIBCXIQVPC-UHFFFAOYSA-N
Compound Name2-isopropoxy-3-(1-((5-methyl-2-(4-(trifluoromethyl)phenyl)oxazol-4-yl)methyl)-1H-indol-5-yl)propanoic acid
Canonical SMILESCc1oc(-c2ccc(C(F)(F)F)cc2)nc1Cn1ccc2cc(CC(OC(C)C)C(=O)O)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.71
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q07869 PPARA Homo sapiens Human PF00104 PF00105 7.2 IC50 ChEMBL;BindingDB
P37231 PPARG Homo sapiens Human PF00104 PF12577 PF00105 6.9 IC50 ChEMBL;BindingDB
Q03181 PPARD Homo sapiens Human PF00104 PF00105 6.0 IC50 ChEMBL;BindingDB