Molecule Details
InChIKeyOZJDKUMSRQSURZ-UHFFFAOYSA-N
Compound Name4-[4-(acetylmethyl-amino)-piperidin-1-yl]-N-(2-chloro-benzyl)-2-(3,4-dichlorophenyl)-2,N-dimethylbutyramide
Canonical SMILESCC(=O)N(C)C1CCN(CCC(C)(C(=O)N(C)Cc2ccccc2Cl)c2ccc(Cl)c(Cl)c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29371 TACR3 Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P25103 TACR1 Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
P21452 TACR2 Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB