Molecule Details
InChIKeyOZGMVFAOJFAKML-UHFFFAOYSA-N
Compound Name1-[3-[3-Ethyl-2-[(3-fluoro-4-pyridinyl)amino]-4-oxothieno[3,2-d]pyrimidin-7-yl]piperidine-1-carbonyl]cyclopropane-1-carbonitrile
Canonical SMILESCCn1c(Nc2ccncc2F)nc2c(C3CCCN(C(=O)C4(C#N)CC4)C3)csc2c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.32
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13946 PDE7A Homo sapiens Human PF00233 9.5 IC50 ChEMBL;BindingDB
Q14432 PDE3A Homo sapiens Human PF00233 7.8 IC50 ChEMBL;BindingDB
Q07343 PDE4B Homo sapiens Human PF18100 PF00233 7.7 IC50 ChEMBL;BindingDB