Molecule Details
InChIKeyOZAXJINUJRJQJM-UHFFFAOYSA-N
Compound Name9-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-1,3-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
Canonical SMILESCOc1ccccc1N1CCN(CCCN2CCCn3c2nc2c3c(=O)n(C)c(=O)n2C)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB