Molecule Details
InChIKeyOYPFBHGNPRGZHS-UHFFFAOYSA-N
Compound Name4-amino-5-cyano-N-(2,5-dimethoxybenzyl)-6-ethoxypyridine-2-carboxamide
Canonical SMILESCCOc1nc(C(=O)NCc2cc(OC)ccc2OC)cc(N)c1C#N
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.75
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.2 IC50 ChEMBL