Target not found.
Molecule Details
InChIKeyOYDMPDMTZYTSSQ-UHFFFAOYSA-N
Compound Nametert-butyl (6-(6-(4-chlorophenyl)-3-cyclopropyl-1-methyl-4-oxopyrrolo[3,4-c]pyrazol-5(1H,4H,6H)-yl)-3-methyl-[1,2,4]triazolo[4,3-a]pyridin-8-yl)carbamate
Canonical SMILESCc1nnc2c(NC(=O)OC(C)(C)C)cc(N3C(=O)c4c(C5CC5)nn(C)c4C3c3ccc(Cl)cc3)cn12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.32
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 7.4 IC50 ChEMBL;BindingDB
P25440 BRD2 Homo sapiens Human PF17035 PF00439 7.3 IC50 ChEMBL;BindingDB
Q15059 BRD3 Homo sapiens Human PF17035 PF00439 7.2 IC50 ChEMBL;BindingDB