Molecule Details
InChIKeyOWIYYKSTVQMPLM-UHFFFAOYSA-N
Compound Name3-Methyl-6-[2-(6-methyl-2-pyridinyl)pyrazol-3-yl]quinazolin-4-one
Canonical SMILESCc1cccc(-n2nccc2-c2ccc3ncn(C)c(=O)c3c2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.56
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P36897 TGFBR1 Homo sapiens Human PF01064 PF00069 PF08515 7.9 IC50 ChEMBL;BindingDB
P36896 ACVR1B Homo sapiens Human PF01064 PF00069 PF08515 7.2 IC50 ChEMBL;BindingDB