Molecule Details
InChIKeyOWHLXTINLAVFEZ-BQYQJAHWSA-N
Canonical SMILESCOc1c(/C=C/c2cc(C(=O)Nc3ccc(CN4CCC(N(C)C)C4)c(C(F)(F)F)c3)ccc2C)cnc2[nH]ccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.22
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P41240 CSK Homo sapiens Human PF07714 PF00017 PF00018 7.6 IC50 ChEMBL
Q16539 MAPK14 Homo sapiens Human PF00069 6.8 IC50 ChEMBL