Molecule Details
InChIKeyOWAPJDQJQMNRHK-UHFFFAOYSA-N
Compound Name2-(3-Amino-6-imino-4,5-disulfoxanthen-9-yl)-5-[6-[4-[4-[[9-chloro-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-yl]amino]-4-oxobutyl]triazol-1-yl]hexylcarbamoyl]benzoic acid
Canonical SMILESN=c1ccc2c(-c3ccc(C(=O)NCCCCCCn4cc(CCCC(=O)Nc5nc6ccc(Cl)cc6c6nc(-c7ccco7)nn56)nn4)cc3C(=O)O)c3ccc(N)c(S(=O)(=O)O)c3oc-2c1S(=O)(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.46
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P0DMS8 ADORA3 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB