Molecule Details
InChIKeyOVXMCCQKIOSDGE-HDICACEKSA-N
Compound Name4-[6-[6-[(2S,6R)-2,6-dimethylpiperazin-1-yl]-3-pyridinyl]pyrazolo[1,5-a]pyrimidin-3-yl]quinoline
Canonical SMILESC[C@@H]1CNC[C@H](C)N1c1ccc(-c2cnc3c(-c4ccnc5ccccc45)cnn3c2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q04771 ACVR1 Homo sapiens Human PF01064 PF07714 PF08515 7.7 IC50 ChEMBL;BindingDB
P37023 ACVRL1 Homo sapiens Human PF07714 PF08515 7.1 IC50 ChEMBL;BindingDB
P36894 BMPR1A Homo sapiens Human PF01064 PF07714 PF08515 7.0 IC50 ChEMBL;BindingDB