Molecule Details
InChIKeyOVNGEJRHHJULAD-AJQTZOPKSA-N
Canonical SMILESCC(C)(C)Oc1cc(C(=O)CC(N)=O)ccc1C1=N[C@@H](c2ccc(C(=O)O)cc2)[C@@H](c2c[nH]c3ccc(Cl)cc23)N1C(=O)N1CCNC(=O)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q00987 MDM2 Homo sapiens Human PF02201 PF13920 PF00641 8.2 IC50 ChEMBL;BindingDB
O15151 MDM4 Homo sapiens Human PF13920 PF00641 7.6 IC50 ChEMBL;BindingDB